D1R agonist | Species | AMPAR current | Result | Neuron Type | Synaptic locus | Region | Reference |
---|---|---|---|---|---|---|---|
SKF 81297 (30 μM) DA (30 μM) | Rat | eEPSC eEPSC, mEPSC | Inhibit // | Magnocellular // | Presynaptic // | BF // | [39] |
SKF 81297 (30 μM) | Rat | eEPSC | Inhibit | Cholinergic | Presynaptic | BF | [40] |
SKF 81297 (1 μM) | Rat | eEPSC | Inhibit | Pyramidal layer V | Presynaptic | PFC | [41] |
SKF 38393 (10 μM) | Rat | eEPSC | Enhance | Pyramidal Layer II/III | Postsynaptic | PFC | [29] |
DA (250 nm-5 μM) | Monkey | eEPSC | Inhibit | Pyramidal layer III | Undetermined | PFC | [42] |
SKF 81297 (1 μM) | Rat | eEPSC | Enhance | Pyramidal Layer II/lll | Postsynaptic | PFC | [43] |
SKF 81297 (5 μM) | Mice | eEPSC | No effect | Pyramidal | – | PFC | [28] |
DA (50 μM) SKF 81297 (10 μM) | Mice // | sEPSC // | Enhance // | D1R+ neurons // | Presynaptic // | Dorsal Striatum // | [44] |
SKF 81297 (1 μM) | Rat | Kainite EPSC |  | Cultured MSN |  | Striatum | [45] |
SKF 38393 (10 M) | Rat | AMPA EPSC | Enhance | MSN | Postsynaptic | Dorsal Striatum | [46] |
SKF 38393 (5 μM) // | Rat // | eEPSC glutamate EPSC | Enhance No effect | MSN // | – – | Striatum | [47] |
DA (75 μM) SKF 81297 (30 μM) SKF 38393 (100 μM) | Rat // // | eEPSP // // | Inhibit No effect LTD | Field & whole cell // // | Presynaptic | NAc // // | [48] |
DA (50 μM) SKF 38393 (10 μM) | Mice | eEPSC // | Inhibit // | MSN // | Postsynaptic // | NAc // | [49] |
SKF 81297 (5 μM) | Mice | Kainate EPSC | enhance | MSN | Postsynaptic | Neostriatum | [50] |
SKF 81297 (5 μM) | Chicken | mEPSC | No effect | Pyramidal layer II/III Motoneurons | – | ACC | [51] |
SKF 38393 (10 μM) | Mice | glutamate EPSC | Enhance |  | – | Embryonic | [52] |