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Table 1 βarrestin2 recruitment to ACKR3-Venus in HEK-293 cells
From:
Ackr3-Venus knock-in mouse lights up brain vasculature
Compound
Emax (%)
LogEC50
CXCL12
100.0 ± 5.6
− 9.15 ± 0.15
VUF11207
73.8 ± 5.6
− 7.78 ± 0.18
TC14012
63.6 ± 4.6
− 6.97 ± 0.14
AMD3100
55.2 ± 6.2
− 7.02 ± 0.23
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